Publications

Found 2 results
Filters: Author is Scholtz, Cole R  [Clear All Filters]
2025
Scholtz, C. R., Doskey, L. C., Kandanur, S. Giridhar S., Vail, N. R., Roderick, E. R., Peterson, E. J., Hoell, Z. J., Shi, K., Aihara, H., Kostallari, E., Shah, V. H., Malhi, H., and Pomerantz, W. C. K. (2025) Development of cell-active BRD4-D1 selective inhibitors to decode the role of BET proteins in LPS-mediated liver inflammation. Eur J Med Chem. 304, 118519
2022
Cui, H., Divakaran, A., Hoell, Z. J., Ellingson, M. O., Scholtz, C. R., Zahid, H., Johnson, J. A., Griffith, E. C., Gee, C. T., Lee, A. L., Khanal, S., Shi, K., Aihara, H., Shah, V. H., Lee, R. E., Harki, D. A., and Pomerantz, W. C. K. (2022) A Structure-based Design Approach for Generating High Affinity BRD4 D1-Selective Chemical Probes. J Med Chem. 10.1021/acs.jmedchem.1c01779